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1-Azakenpaullone

抑制糖原合成酶激酶3β (GSK3β)

产品号 #(选择产品)

产品号 #74252_C

抑制糖原合成酶激酶3β (GSK3β)

总览

1-Azakenpaullone 是一种强效且高选择性的糖原合酶激酶 3β (IC₅₀ = 18 nM) 抑制剂,并且相对于其他细胞周期依赖性激酶 (CDK),包括 CDK/细胞周期蛋白 B 和 CDK5/p25  (IC₅₀ = 2 µM and 4.2 µM, respectively; Kunick et al.),其对 GSK3β 的作用更佳。


维持和自我更新
·与ID-8(产品号 #72502)和FK506(产品号 #74152)联合使用,可支持人多能干细胞的长期增殖、维持多能性和分化能力(Yasuda et al.)。

细胞类型
多能干细胞
 
种属
人,小鼠,非人灵长类,其它细胞系,大鼠
 
应用
培养
 
研究领域
干细胞生物学
 
CAS 编号
676596-65-9
 
化学式
C₁₅H₁₀BrN₃O
 
纯度
≥98%
 
靶点
GSK3β
 

Protocols and Documentation

Find supporting information and directions for use in the Product Information Sheet or explore additional protocols below.

Document Type
Product Name
Catalog #
Lot #
Language
Product Name
1-Azakenpaullone
Catalog #
74252
Lot #
All
Language
English
Document Type
Safety Data Sheet
Product Name
1-Azakenpaullone
Catalog #
74252
Lot #
All
Language
English

Applications

This product is designed for use in the following research area(s) as part of the highlighted workflow stage(s). Explore these workflows to learn more about the other products we offer to support each research area.

更多信息

更多信息
种属 Human, Mouse, Non-Human Primate, Other, Rat
Cas Number 676596-65-9
Chemical Formula C₁₅H₁₀BrN₃O
纯度 ≥ 98%
Target GSK3β
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